Various inhibitors and other biologically active compounds
OTAVA has extensive experience in the synthesis of highly valuable products for biotech and pharmaceutical applications around the world.

Our company offers a number of INHIBITORS and other biologically active compounds modulating activity of distinct targets (see below). These compounds are available in milligram and gram quantities. Custom and bulk quotes are also available. Please contact us for quotes.

If you do not see a compound you are looking for, we offer Custom Synthesis Services. Please contact us for quotes and details.



Download ALL in ONE file:  Bioactive Small Molecules Catalog (2012)

 

Biological activity

OTAVA catalog no.

CAS RN

Product sheet

SIRT1 activator

1091797

374922-43-7

 Read more

CINK4 - Cdk4/6 Inhibitor IV

1112092

359886-84-3

 Read more

CP-547632 - VEGFR-2 and FGFR1 inhibitor

1156353

252003-65-9

 Read more

Cediranib ( AZD2171 ) – VEGFR inhibitor

1156354

288383-20-0

 Read more

Vandetanib (ZD6474; Zactima ) – VEGFR and EGFR inhibitor

1156355

443913-73-3

 Read more

VEGFR-2 inhibitor

1156358

769960-39-6

 Read more

Inhibitor of the Hedgehog Signalling Pathway

1156359

330796-24-2

Read more

NSC 702827 (SU 6668; TSU 68) - PDGFR, VEGFR and FGFR inhibitor

1156360

252916-29-3

 Read more

ARRY 142886 (AZD 6244) - Mitogen-activated protein kinase 1/2 inhibitor

1183194

606143-52-6

Read more

SK&F 29661 - Inhibitor of Phenylethanolamine N-Methyl-Transferase

1183326

31404-61-2

 Read more

iso-AZD6244 (avialable eclusively from Otava)

1901577

N/A

 Read more

CK2 inhibitor

0107830107

300675-28-9

Read more

CK2 inhibitor

0107830108

302553-01-1

 Read more

NSC 210902 – CK2 inhibitor

0107830116

51726-83-1

 Read more

AGK-2 - SIRT2 Inhibitor

0117392020

304896-28-4

Read more

CFTRinh-172 - Voltage-independent, selective CFTR chloride channel blocker

0129690030

307510-92-5

 Read more

Inhibitor of the deubiquitinating activity of human USP14

0129720262

314245-33-5

Read more

Janex 3 (WHI-P180) - Cyclin-dependent Kinase (CDK) Inhibitor

7015070102

211555-08-7

 Read more

Janex-1 ( WHI-P131 ) - Janus kinase 3 inhibitor

7015070103

202475-60-3

 Read more

CK2 inhibitor

7015980251

19231-60-8

 Read more

EX-527 - Inhibitor of the deacetylase SIRT1

7020402314

49843-98-3

 Read more 

Cambinol ( NSC-112546 ) - SIRT1/2 Inhibitor IV

7020402315

14513-15-6

 Read more

IQA (CGP029482) - CK2 inhibitor

7020402316

391670-48-7

 Read more

CAN508 - CDK9 Inhibitor II

7020402317

140651-18-9

 Read more

Polo-like kinase 1 (PLK1) inhibitor

7020402323

916985-21-2

 Read more

Inhibitor of IKK- ε kinase

7020402324

862812-98-4

 Read more

Inhibitor of cGMP-specific phosphodiesterase

7020540496

150450-42-3

 Read more

AG 1517 (NSC669364; PD 153035; SU 5271; WHI-P79) - EGFR-kinase inhibitor

7020540711

153436-54-5

 Read more

ZXX2-77 - Benzenesulfonanilide-type cyclooxygenase-1-selective inhibitor

7070707001

304913-22-2

 Read more

GW1100 - GPR40 antagonist

7070707009

306974-70-9

 Read more

4EGI- 1 - eIF4E/eIF4G Interaction Inhibitor

7070707011

315706-13-9

 Read more

NH125 - eEF-2 Kinase Inhibitor

7070707012

278603-08-0

 Read more

TWS119 - Glycogen synthase kinase-3 (GSK-3) inhibitor

7070707013

601514-19-6

 Read more

Antagonist of NMDA receptor

7070707014

81094-64-6

 Read more

LW6 - Hypoxia Inducible Factor-1α Inhibitor

7070707015

934593-90-5

Read more

HNHA - Histone Deacetylase Inhibitor VI

7070707016

926908-04-5

 Read more

IQ-1 - Stem Cell Reagent; Wnt Pathway Activator III

7070707017

331001-62-8

 Read more

NSC 74859 (S3I-201)) - STAT3 Inhibitor VI

7070707021

501919-59-1

 Read more

Compound 401 - Selective DNA-PK and mTOR inhibitor

7070707024

168425-64-7

 Read more

A-769662 - AMPK activator

7070707027

844499-71-4

Read more

PIK-90 - PI3K Inhibitor

7070707028

677338-12-4

Read more

PIK-93 - PI4-kinase inhibitor

7070707029

593960-11-3

Read more

Bifeprunox - Partial dopamine D2 agonist; 5-HT1A agonist

7070707030

350992-10-8

 Read more

cFMS Receptor Tyrosine Kinase Inhibitor

7070707032

959626-45-0

 Read more

Cdk4 Inhibitor

7070707035

546102-60-7

 Read more

PD166866 - Inhibitor of basic Fibroblast Growth Factor (bFGF)

7070707041

192705-79-6

 Read more

BX-795 - PDK1 inhibitor

7070707044

702675-74-9

 Read more

BX-320 - PDK1 inhibitor

7070707045

702676-93-5

 Read more

IC87114 - Inhibitor of the p110δ isoform of PI3 kinase

7070707046

371242-69-2

Read more

TGX155 - PI3K Inhibitor

7070707047

351071-90-4

 Read more

R112 - Syk kinase inhibitor

7070707049

575474-82-7

 Read more

OSU03012 - PDK1 Inhibitor

7070707053

742112-33-0

 Read more

Syk kinase inhibitor

7070707056

726695-51-8

 Read more

WP1066 - JAK2 Inhibitor

7070707057

857064-38-1

 Read more

TGX115 - Inhibitor of PI3 kinase

7070707058

351071-62-0

 Read more

BX-912 - PDK1 inhibitor

7070707060

702674-56-4

 Read more

PD-0325901 - Mitogenic extracellular kinase 1/2 (MEK1/2) inhibitor

7070707062

391210-10-9

 Read more

WAY-265497 - Cdk4 Inhibitor

7070707068

943746-57-4

 Read more

SU 3327 - inhibitor of c-Jun N-terminal kinase

7070707069

40045-50-9

 Read more

Inhibitor of Nek2/Hec1

7070707071

1001753-24-7

 Read more

Inhibitor of Nek2/Hec1

7070707072

560103-80-2

Read more

HDAC1 & 2 Inhibitor

7070707089

1013330-84-1

 Read more

HDAC1 & 2 Inhibitor

7070707091

849234-64-6

 Read more

Thiazovivin - Cell survival promoting small molecule

7070707131

1226056-71-8

 Read more

BRAF Inhibitor

7070707132

884339-61-1

 Read more

NSC109116 - Human 20α-hydroxysteroid dehydrogenase (AKR1C1) inhibitor

7070707133

4906-68-7

Read more

VUF 8430 - Histamine H4 receptor agonist

7070707134

100130-32-3

 Read more

Arcyriaflavin A - Cdk4 Inhibitor

7070707137

118458-54-1

 Read more

ATBAC (C-3; C-Tre; Capobenic acid; NSC230936; TB-ACA) - Cardial depressant (antiarrhythmic)

7110950124

21434-91-3

Read more

VU0155041 - Potent and positive allosteric mGlu4 agonist

7114471128

1093757-42-6

 Read more

PAC-1 - Antitumor agent activating procaspase-3 to caspase-3

7210801533

315183-21-2

Read more

STF-62247 - Autophagy Inducer

7211760086

315702-99-9

 Read more

JK 184 - Inhibitor of the Hedgehog Signalling Pathway

7211760148

315703-52-7

 Read more

Tenovin 1 - p53 activator

7215270035

380315-80-0

 Read more
Dual PI3K-α and mTOR inhibitor 7070707142 1197160-78-3 Read more
Dual VEGFR-2 and tubulin inhibitor 7070707143 830333-53-4 Read more
HDAC, EGFR, and HER2 inhibitor 7070707144 1012054-55-5 Read more

VEGFR Inhibitor

7070707147

690206-97-4

Read more

ROCK Inhibitor

7070707146

1225199-26-7

Read more

mTOR inhibitor (Torin2)

7070707148

1223001-51-1

Read more

K-604, selective ACAT-1 inhibitor

7070707145

561023-90-3

Read more

TCS 21311, selective JAK3 inhibitor

7070707149

1260181-14-3

Read more

New Protein kinase CK2 inhibitor (available exclusively from Otava)

1436838

1181227-92-8

Read more

New inhibitor of the human protein kinase CK2 (available exclusively from Otava)

1234350

329907-28-0

Read more

New inhibitor of human protein kinase ASK1 (MAP3K5, MAPKKK5, MEKK5) (available exclusively from Otava)

7214191049

175026-96-7

Read more

Nitric oxide synthase (inducible) Inhibitor

1055516

1532-84-9

Read more

Inhibitor of erbB1 and p56lck

7020540710

N/A

Read more

Inhibitor of EGFR

7020540007

N/A

Read more

Inhibitor of monoamine oxidase (MAO) and aldehyde dehydrogenase (ALDH-2)

7119860038

486-66-8

Read more

Inhibitor of protein kinase ABL

7119681298

N/A

Read more

Inhibitor of Hepatitis C virus NS3 protease/helicase

7119561895

85-55-2

Read more

EGFR  Inhibitor

7017500003

N/A

Read  more

EGFR  Inhibitor

7017500002

N/A

Read more

EGFR Inhibitor

7017500001

N/A

Read more

Beta amyloid A4 protein Inhibitor

7216513379

6278-73-5

Read more

EGFR Inhibitor

7015070078

N/A

Read more

Inhibitor of MAO-A and MAO-B

7113231449

N/A

Read more

Kinesin-like protein 1 Inhibitor

7112880116

N/A

Read more

Inhibitor of MAO-B and MAO-A

7012702160

N/A

Read more

Inhibitor of valosin-containing protein (VCP or p97)

7211760421

312636-16-1

Read more

Inhibitor of valosin-containing protein (VCP or p97)

7211760110

N/A

Read more

EGFR Inhibitor

7011830583

N/A

Read more

Inhibitor of MAO-A and MAO-B

7210430507

307548-94-3

Read more

EGFR Inhibitor

0108440188

N/A

Read more

EGFR Inhibitor

0108440177

N/A

Read more

EGFR Inhibitor

0108440173

N/A

Read more

EGFR Inhibitor

0108440170

N/A

Read more

EGFR Inhibitor

0108440152

N/A

Read more

EGFR Inhibitor

0107930017

6178-42-3

Read more

Carbonic anhydrase IX Inhibitor

0127441873

N/A

Read more

Protein kinase ABL Inhibitor

0117391283

N/A

Read more

Hepatitis C virus NS3 protease/helicase inhibitor

0125160292

496-41-3

Read more

EGFR Inhibitor

0116690044

5334-30-5

Read more

hMAO-B and hMAO-A Inhibitor

0105860050

N/A

Read more

hMAO-A and hMAO-B Inhibitor

0115540187

N/A

Read more

hMAO-A and hMAO-B Inhibitor

0115540186

N/A

Read more

Inhibitor of MAO-B and MAO-A

0115540181

N/A

Read more

MAO B Inhibitor

0115540179

N/A

Read more

MAO B Inhibitor

0115540178

N/A

Read more

Serine/threonine-proteine kinase PIM1/PIM2 Inhibitor

0123300047

N/A

Read more

MAO B Inhibitor

5030790694

N/A

Read more
Need more information regarding this product? Send us an inquiry:


Name: *
Company: *
E-mail: *
Your message
(please specify name of the product
you are interested in):
*
Word Verification: