 GPCR Agonists Focused Library The library has the following predicted activities: • 5 Hydroxytryptamine agonist • Acetylcholine muscarinic agonist • Alpha adrenoreceptor agonist • Beta adrenoreceptor agonist • Cholecystokinin agonist • Dopamine agonist • Dopamine autoreceptor agonist • GABA receptor agonist • Melatonin agonist Additional Details: - Number of compounds in library: ~ 460
- Preparation method: SAR
Feel free to contact us if you are interested to obtain these libraries or if you need extra information.
GPCR Antagonists Focused Library The library has the following predicted activities: • 5 Hydroxytryptamine antagonist • Acetylcholine muscarinic antagonist • Adenosine receptor antagonist • Alpha adrenoreceptor antagonist • Beta adrenoreceptor antagonist • Dopamine antagonist • Endothelin receptor antagonist • GABA receptor antagonist • Glucagon receptor antagonist • Glutamate receptor antagonist • Histamine antagonist • Melatonin antagonist • Neuropeptide antagonist • Prostaglandin antagonist • Thromboxane antagonist • Vasopressin 1 antagonist Additional Details: Feel free to contact us if you are interested to obtain these libraries or if you need extra information.
Protein Kinase Inhibitors Focused Library The library has the following predicted activities: • 1-Phosphatidylinositol-4-phosphate 5-kinase inhibitor • Abl kinase inhibitor • Acetate kinase inhibitor • ADP-thymidine kinase inhibitor • Aurora kinase inhibitor • Aurora-B kinase inhibitor • Aurora-C kinase inhibitor • Beta-adrenergic receptor kinase inhibitor • Check point kinase inhibitor • Cyclin-dependent kinase 1 inhibitor • Cyclin-dependent kinase 2 inhibitor • Cyclin-dependent kinase 4 inhibitor • Cyclin-dependent kinase inhibitor • EphB2 kinase inhibitor • Epidermal growth factor receptor kinase inhibitor • Glycogen synthase kinase-3 inhibitor • G-protein-coupled receptor kinase inhibitor • Guanidinoacetate kinase inhibitor • I kappa B kinase 2 inhibitor • Inositol-trisphosphate 3-kinase inhibitor • Lombricine kinase inhibitor • MAP kinase inhibitor • N-acylmannosamine kinase inhibitor • NADH kinase inhibitor • Opheline kinase inhibitor • Phosphatidylinositol 3-kinase beta inhibitor • Phosphatidylinositol 3-kinase gamma inhibitor • Phosphoenolpyruvate carboxykinase (diphosphate) inhibitor • Platelet derived growth factor receptor kinase inhibitor • Protein kinase (CK1) inhibitor • Protein kinase B inhibitor • Protein kinase C eta inhibitor • Protein-serine-threonine kinase inhibitor • Proto-oncogene tyrosine-protein kinase Fyn inhibitor • Proto-oncogene tyrosine-protein kinase Kit inhibitor • Pyridoxal kinase inhibitor • Raf kinase B inhibitor • Raf kinase inhibitor • Rho-associated kinase inhibitor • Ribosomal protein S6 kinase inhibitor • Shikimate kinase inhibitor • Smooth muscle myosin light chain kinase inhibitor • Sphinganine kinase inhibitor • Sphingosine kinase inhibitor • Src kinase inhibitor • Taurocyamine kinase inhibitor • Thymidine kinase inhibitor • Tyrosine kinase inhibitor • Urokinase inhibitor Additional Details: Feel free to contact us if you are interested to obtain these libraries or if you need extra information.
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