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Protein families libraries

f_libraries.jpgarrow_bullet.gifGPCR Agonists Focused Library

The library has the following predicted activities:

• 5 Hydroxytryptamine agonist
• Acetylcholine muscarinic agonist
• Alpha adrenoreceptor agonist
• Beta adrenoreceptor agonist
• Cholecystokinin agonist
• Dopamine agonist
• Dopamine autoreceptor agonist
• GABA receptor agonist
• Melatonin agonist

Additional Details:

  • Number of compounds in library: ~ 460
  • Preparation method: SAR

 


Feel free to contact us if you are interested to obtain these libraries or if you need extra information.




arrow_bullet.gifGPCR Antagonists Focused Library

The library has the following predicted activities:

• 5 Hydroxytryptamine antagonist
• Acetylcholine muscarinic antagonist
• Adenosine receptor antagonist
• Alpha adrenoreceptor antagonist
• Beta adrenoreceptor antagonist
• Dopamine antagonist
• Endothelin receptor antagonist
• GABA receptor antagonist
• Glucagon receptor antagonist
• Glutamate receptor antagonist
• Histamine antagonist
• Melatonin antagonist
• Neuropeptide antagonist
• Prostaglandin antagonist
• Thromboxane antagonist
• Vasopressin 1 antagonist

Additional Details:

  • Number of compounds in library: ~ 4900
  • Preparation method: SAR

 


Feel free to contact us if you are interested to obtain these libraries or if you need extra information.




arrow_bullet.gifProtein Kinase Inhibitors Focused Library

The library has the following predicted activities:

• 1-Phosphatidylinositol-4-phosphate 5-kinase inhibitor
• Abl kinase inhibitor
• Acetate kinase inhibitor
• ADP-thymidine kinase inhibitor
• Aurora kinase inhibitor
• Aurora-B kinase inhibitor
• Aurora-C kinase inhibitor
• Beta-adrenergic receptor kinase inhibitor
• Check point kinase inhibitor
• Cyclin-dependent kinase 1 inhibitor
• Cyclin-dependent kinase 2 inhibitor
• Cyclin-dependent kinase 4 inhibitor
• Cyclin-dependent kinase inhibitor
• EphB2 kinase inhibitor
• Epidermal growth factor receptor kinase inhibitor
• Glycogen synthase kinase-3 inhibitor
• G-protein-coupled receptor kinase inhibitor
• Guanidinoacetate kinase inhibitor
• I kappa B kinase 2 inhibitor
• Inositol-trisphosphate 3-kinase inhibitor
• Lombricine kinase inhibitor
• MAP kinase inhibitor
• N-acylmannosamine kinase inhibitor
• NADH kinase inhibitor
• Opheline kinase inhibitor
• Phosphatidylinositol 3-kinase beta inhibitor
• Phosphatidylinositol 3-kinase gamma inhibitor
• Phosphoenolpyruvate carboxykinase (diphosphate) inhibitor
• Platelet derived growth factor receptor kinase inhibitor
• Protein kinase (CK1) inhibitor
• Protein kinase B inhibitor
• Protein kinase C eta inhibitor
• Protein-serine-threonine kinase inhibitor
• Proto-oncogene tyrosine-protein kinase Fyn inhibitor
• Proto-oncogene tyrosine-protein kinase Kit inhibitor
• Pyridoxal kinase inhibitor
• Raf kinase B inhibitor
• Raf kinase inhibitor
• Rho-associated kinase inhibitor
• Ribosomal protein S6 kinase inhibitor
• Shikimate kinase inhibitor
• Smooth muscle myosin light chain kinase inhibitor
• Sphinganine kinase inhibitor
• Sphingosine kinase inhibitor
• Src kinase inhibitor
• Taurocyamine kinase inhibitor
• Thymidine kinase inhibitor
• Tyrosine kinase inhibitor
• Urokinase inhibitor

Additional Details:

  • Number of compounds in library: ~ 10,000
  • Preparation method: SAR

 


Feel free to contact us if you are interested to obtain these libraries or if you need extra information.