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All Focused Libraries

Full list of Focused LibrariesFull collection of more than  350 OTAVAchemicals's Focused Libraries designed with Receptor-based or Ligand-based approach is represented here.

These libraries are proposed for screening in various research and drug development projects.

 

 

 

 

 

  • the libraries contain drug-like compounds only
  • all the compounds are in stock
  • cherry picking is available

 

You can sort data by any column and use "Filter" option to search library's name:

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Name Number of compounds Approach Details
1-Phosphatidylinositol-4-phosphate 5-kinase (PIPK) inhibitor 14 Ligand-based -
Abl kinase inhibitor 76 Ligand-based -
Acetate kinase inhibitor 129 Ligand-based -
ADP-thymidine kinase inhibitor 922 Ligand-based -
Aurora kinase inhibitor 364 Ligand-based -
Aurora-B kinase inhibitor 249 Ligand-based -
Aurora-C kinase inhibitor 1162 Ligand-based -
Beta-adrenergic receptor kinase (BARK) inhibitor 1268 Ligand-based -
Check point kinase (CHK) inhibitor 593 Ligand-based -
Cyclin-dependent kinase 1 (CDK1) inhibitor 83 Ligand-based -
Cyclin-dependent kinase 2 (CDK2) inhibitor 905 Ligand-based -
Cyclin-dependent kinase 4 (CDK4) inhibitor 798 Ligand-based -
Cyclin-dependent kinase (CDK) inhibitor 285 Ligand-based -
EphB2 kinase inhibitor 329 Ligand-based -
Epidermal growth factor receptor kinase (EGFR) inhibitor 318 Ligand-based -
Glycogen synthase kinase-3 (GSK3) inhibitor 153 Ligand-based -
G-protein-coupled receptor kinase (GRK) inhibitor 1268 Ligand-based -
Guanidinoacetate kinase inhibitor 254 Ligand-based -
I kappa B kinase 2 (IKK2) inhibitor 347 Ligand-based -
Inositol-trisphosphate 3-kinase (IP3K) inhibitor 78 Ligand-based -
Lombricine kinase inhibitor 163 Ligand-based -
MAP kinase (MAPK) inhibitor 102 Ligand-based -
N-acylmannosamine kinase inhibitor 935 Ligand-based -
NADH kinase inhibitor 871 Ligand-based -
Opheline kinase inhibitor 875 Ligand-based -
Phosphatidylinositol 3-kinase beta (PI3K-C2 beta) inhibitor 1183 Ligand-based -
Phosphatidylinositol 3-kinase gamma (PI3K-C2 gamma) inhibitor 252 Ligand-based -
Phosphoenolpyruvate carboxykinase (PEPCK) inhibitor 26 Ligand-based -
Platelet derived growth factor receptor kinase (PDGFR) inhibitor 1972 Ligand-based -
Protein kinase CK1 inhibitor 1387 Ligand-based -
Protein kinase B (PKB) inhibitor 1030 Ligand-based -
Protein kinase C eta (PKC) inhibitor 16 Ligand-based -
Protein-serine-threonine kinase inhibitor 213 Ligand-based -
Proto-oncogene tyrosine-protein kinase Fyn inhibitor 481 Ligand-based -
Proto-oncogene tyrosine-protein kinase Kit inhibitor 214 Ligand-based -
Pyridoxal kinase inhibitor 5 Ligand-based -
Raf kinase B inhibitor 38 Ligand-based -
Raf kinase inhibitor 74 Ligand-based -
Rho-associated kinase inhibitor 344 Ligand-based -
Ribosomal protein S6 kinase (S6K) inhibitor 10 Ligand-based -
Shikimate kinase inhibitor 453 Ligand-based -
Smooth muscle myosin light chain kinase (MLCK) inhibitor 627 Ligand-based -
Sphinganine kinase inhibitor 244 Ligand-based -
Sphingosine kinase inhibitor 1119 Ligand-based -
Src kinase inhibitor 200 Ligand-based -
Taurocyamine kinase inhibitor 875 Ligand-based -
Thymidine kinase inhibitor 922 Ligand-based -
Tyrosine kinase inhibitor 1147 Ligand-based -
Urokinase inhibitor 21 Ligand-based -
P21-Activated Kinase 1 (PAK1) 2024 Receptor-based read more
Serine/Threonine-Protein Kinase CHK1 (CHK1) 1946 Receptor-based read more
Proto-Oncogene Tyrosine-Protein Kinase ABL1 2048 Receptor-based read more
Extracellular Signal-Regulated Kinase 2 (ERK2) 2053 Receptor-based read more
Death-Associated Protein Kinase 2 (DAPK-2) 2012 Receptor-based read more
p38 MAP Kinase Alpha 2221 Receptor-based read more
Vascular Endothelial Growth Factor Receptor 2 (VEGFR2) 2235 Receptor-based read more
Aurora B kinase 2069 Receptor-based read more
Janus Kinase 2 (Jak2) 2190 Receptor-based read more
Phosphatidylinositol 3-kinase (PI3K) 2040 Receptor-based read more
3-phosphoinositide-dependent kinase-1 (PDK-1) 1975 Receptor-based read more
Cyclin Dependent Kinase 2 (CDK2) 1281 Receptor-based read more
Glycogen Synthase Kinase-3 (GSK3) 980 Receptor-based read more
Fibroblast growth factor receptor 1 tyrosine kinase (FGFR1K) 1761 Receptor-based read more
cAMP dependent protein kinase (PKA) 1877 Receptor-based read more
C-Jun N-Terminal Kinase 2 (Jnk2, Mapk9) 1774 Receptor-based -
Death-associated protein kinase 1 (DAPK1) 1962 Receptor-based -
Death-associated protein kinase 3 (DAPK3) 1814 Receptor-based -
DOT1-like, histone H3 methyltransferase (DOT1L) inhibitors 670 Receptor-based read more
Bromodomain-containing protein 4 (BRD4) inhibitors 370 Receptor-based read more
Histone Deacetylase (HDAC) inhibitors 947 Receptor-based read more
DNA (cytosine-5)-methyltransferase 1 (DNMT1) inhibitors 503 Receptor-based read more
DNA (cytosine-5)-methyltransferase 3 beta (DNMT3b) inhibitors 1320 Receptor-based read more
Histone Acetyltransferase (HAT) inhibitors 859 Receptor-based read more
CREB binding protein (CREBBP) 664 Receptor-based read more
Angiogenesis inhibitor 1625 Ligand-based -
Antipsychotic 1315 Ligand-based -
Antiobesity 1714 Ligand-based -
Antimigraine 426 Ligand-based -
Antidepressant 1554 Ligand-based -
Anticonvulsant 1830 Ligand-based -
Anticarcinogenic 822 Ligand-based -
Antifungal 828 Ligand-based -
Antimycobacterial 1696 Ligand-based -
Antituberculosic 1828 Ligand-based -
Acaricide - Ligand-based -
Adrenergic - Ligand-based -
Adrenergic, ophthalmic - Ligand-based -
Analeptic - Ligand-based -
Analgesic - Ligand-based -
Analgesic, non-opioid - Ligand-based -
Anesthetic - Ligand-based -
Anesthetic general - Ligand-based -
Anesthetic inhalation - Ligand-based -
Anesthetic local - Ligand-based -
Anorexic - Ligand-based -
Antiadrenergic - Ligand-based -
Antiallergic - Ligand-based -
Antiamebic - Ligand-based -
Antianginal - Ligand-based -
Antiarrhythmic - Ligand-based -
Antibacterial - Ligand-based -
Anticataract - Ligand-based -
Anticoagulant - Ligand-based -
Antidiabetic - Ligand-based -
Antidiabetic symptomatic - Ligand-based -
Antiglaucomic - Ligand-based -
Antihelmintic - Ligand-based -
Antihistaminic - Ligand-based -
Antihypercholesterolemic - Ligand-based -
Antihypertensive - Ligand-based -
Antiinfective - Ligand-based -
Antiinflammatory - Ligand-based -
Antiinflammatory, intestinal - Ligand-based -
Antiischemic, cerebral - Ligand-based -
Antineoplastic - Ligand-based -
Antineoplastic enhancer - Ligand-based -
Antiosteoporotic - Ligand-based -
Antioxidant - Ligand-based -
Antiparasitic - Ligand-based -
Antiparkinsonian - Ligand-based -
Antiprotozoal - Ligand-based -
Antiprotozoal (Coccidial) - Ligand-based -
Antipsoriatic - Ligand-based -
Antipyretic - Ligand-based -
Antischistosomal - Ligand-based -
Antisecretoric - Ligand-based -
Antiseptic - Ligand-based -
Antithrombotic - Ligand-based -
Antitreponemal - Ligand-based -
Antitrypanosomal - Ligand-based -
Antitussive - Ligand-based -
Antiulcerative - Ligand-based -
Antiuremic - Ligand-based -
Antiviral - Ligand-based -
Anxiolytic - Ligand-based -
Bone diseases treatment - Ligand-based -
Bone formation stimulant - Ligand-based -
Bronchodilator - Ligand-based -
Capillary fragility treatment - Ligand-based -
Carcinogenic - Ligand-based -
Cardiodepressant - Ligand-based -
Cardiotonic - Ligand-based -
Choleretic - Ligand-based -
Cholesterol synthesis inhibitor - Ligand-based -
Cholinergic - Ligand-based -
Cholinergic antagonist - Ligand-based -
CNS active muscle relaxant - Ligand-based -
Coagulant - Ligand-based -
Cognition disorders treatment - Ligand-based -
Cytostatic - Ligand-based -
Dermatologic - Ligand-based -
Diuretic - Ligand-based -
Diuretic inhibitor - Ligand-based -
DNA synthesis inhibitor - Ligand-based -
Embryotoxic - Ligand-based -
Expectorant - Ligand-based -
Free radical scavenger - Ligand-based -
Growth stimulant - Ligand-based -
Hemostatic - Ligand-based -
Hepatic disorders treatment - Ligand-based -
Hepatoprotectant - Ligand-based -
Hypertensive - Ligand-based -
Hypoglycemic - Ligand-based -
Hypolipemic - Ligand-based -
Hypotermic - Ligand-based -
Insecticide - Ligand-based -
Insulin secretagoues - Ligand-based -
Keratolytic - Ligand-based -
Miotic - Ligand-based -
Muscle relaxant - Ligand-based -
Mutagenic - Ligand-based -
Oxytocic - Ligand-based -
Protein synthesis inhibitor - Ligand-based -
Psychotropic - Ligand-based -
Radioprotector - Ligand-based -
Radiosensitizer - Ligand-based -
Reductant - Ligand-based -
Renal disease treatment - Ligand-based -
Respiratory analeptic - Ligand-based -
Restenosis treatment - Ligand-based -
Saluretic - Ligand-based -
Sedative - Ligand-based -
Skeletal muscle relaxant - Ligand-based -
Skin irritative effect - Ligand-based -
Sleep disorders treatment - Ligand-based -
Spasmogenic - Ligand-based -
Spasmolytic - Ligand-based -
Spasmolytic, Papaverin-like - Ligand-based -
Spasmolytic, urinary - Ligand-based -
Sweetener - Ligand-based -
Teratogen - Ligand-based -
Ulcerogenic - Ligand-based -
Uric acid diuretic - Ligand-based -
Uricosuric - Ligand-based -
Urinary incontinence treatment - Ligand-based -
Uterine relaxant - Ligand-based -
Vasodilator - Ligand-based -
Vasodilator, coronary - Ligand-based -
Antiviral (hepatitis C) - Ligand-based -
Antiviral (hepatitis) - Ligand-based -
Antiviral (poxvirus) - Ligand-based -
Antiviral (trachoma) - Ligand-based -
GPCR Agonists 465 Ligand-based -
5 Hydroxytryptamine agonist 54 Ligand-based -
Acetylcholine muscarinic agonist 10 Ligand-based -
Alpha adrenoreceptor agonist 45 Ligand-based -
Cholecystokinin agonist 12 Ligand-based -
Dopamine agonist 29 Ligand-based -
Dopamine autoreceptor agonist 181 Ligand-based -
GABA receptor agonist 117 Ligand-based -
Melatonin agonist 17 Ligand-based -
GPCR Antagonists 5089 Ligand-based -
5 Hydroxytryptamine antagonist 347 Ligand-based -
Acetylcholine muscarinic antagonist 81 Ligand-based -
Adenosine receptor antagonist 110 Ligand-based -
Alpha adrenoreceptor antagonist 1045 Ligand-based -
Beta adrenoreceptor antagonist 89 Ligand-based -
Dopamine antagonist 61 Ligand-based -
Endothelin receptor antagonist 165 Ligand-based -
GABA receptor antagonist 1133 Ligand-based -
Glucagon receptor antagonist 526 Ligand-based -
Glutamate receptor antagonist 15 Ligand-based -
Histamine antagonist 590 Ligand-based -
Neuropeptide antagonist 106 Ligand-based -
Prostaglandin antagonist 665 Ligand-based -
Thromboxane antagonist 133 Ligand-based -
Vasopressin 1 antagonist 23 Ligand-based -
5-Hydroxytryptamine Receptor (5-HT1B) Antagonist 1836 Receptor-based read more
Histamine Receptor Antagonist 1295 Receptor-based read more
Hyperpolarization-Activated Cyclic Nucleotide-Gated (HCN) Channel Blocker 765 Ligand-based read more
Calcium Channel Blockers 1262 Ligand-based read more
Calcium Channel Antagonist 165 Ligand-based -
Sodium Channel Blocker 1281 Ligand-based -
Voltage-gated sodium channel blocker 1630 Ligand-based read more
Kv1.5 potassium channel blocker 1052 Ligand-based read more
Glucocorticoid Receptor Antagonist library 1600 Receptor-based read more
Liver X Receptor beta modulator 560 Receptor-based read more
Trypsin inhibitor 85 Ligand-based -
Factor Xa inhibitor 122 Ligand-based -
Tryptase inhibitor 139 Ligand-based -
Cathepsin B inhibitor 275 Ligand-based -
Cathepsin L inhibitor 71 Ligand-based -
Cathepsin T inhibitor 1550 Ligand-based -
Subtilisin inhibitor 123 Ligand-based -
HCV serine protease inhibitor 1300 Ligand-based -
Matrix metalloproteinase 1 inhibitor 39 Ligand-based -
Matrix metalloproteinase inhibitor 16 Ligand-based -
Metalloproteinase inhibitor 21 Ligand-based -
Metalloproteinase-9 inhibitor 608 Ligand-based -
Glycomimetic 246 Ligand-based read more
Beta-turn Peptidomimetic Library 520 Ligand-based read more
Protein-protein interactions (PPI) inhibitor iPPI Tree 1330 Ligand-based read more
Protein-protein interactions (PPI) inhibitor iPPI Bayesian 2310 Ligand-based read more
RNA targeted library - Ligand-based read more
DPP4 focused library 740 Ligand-basedReceptor-based read more
RNA targeted library 3065 Ligand-based read more
Acetylcholine M2 receptor antagonist - Ligand-based -
Acetylcholine M3 receptor antagonist - Ligand-based -
Acetylcholinesterase (AChE) 828 Receptor-based -
Acetylcholine muscarinic antagonist - Ligand-based -
Alpha 1 adrenoreceptor agonist - Ligand-based -
Alpha 1 adrenoreceptor antagonist - Ligand-based -
Alpha 1a adrenoreceptor antagonist - Ligand-based -
Alpha 2 adrenoreceptor agonist - Ligand-based -
Alpha adrenoreceptor agonist - Ligand-based -
Alpha adrenoreceptor antagonist - Ligand-based -
Dopamine autoreceptor agonist - Ligand-based -
Dopamine D3 agonist - Ligand-based -
Dopamine D3 antagonist - Ligand-based -
Dopamine D4 antagonist - Ligand-based -
Endothelin A receptor antagonist - Ligand-based -
Endothelin B receptor antagonist - Ligand-based -
Endothelin receptor antagonist - Ligand-based -
GABA A receptor agonist - Ligand-based -
Glucagon receptor antagonist - Ligand-based -
2,3 Oxidosqualene lanosterol cyclase inhibitor - Ligand-based -
5 Hydroxytryptamine 1 antagonist - Ligand-based -
5 Hydroxytryptamine 1A agonist - Ligand-based -
5 Hydroxytryptamine 1D antagonist - Ligand-based -
5 Hydroxytryptamine 2 agonist - Ligand-based -
5 Hydroxytryptamine 2A antagonist - Ligand-based -
5 Hydroxytryptamine 2C antagonist - Ligand-based -
5 Hydroxytryptamine 3 agonist - Ligand-based -
5 Hydroxytryptamine antagonist - Ligand-based -
5 Hydroxytryptamine uptake inhibitor - Ligand-based -
Acetyl CoA transferase inhibitor - Ligand-based -
Acetylcholine nicotinic agonist - Ligand-based -
Acetylcholine nicotinic antagonist - Ligand-based -
Acute neurologic disorders treatment - Ligand-based -
ADP ribose polymerase inhibitor - Ligand-based -
Adrenaline antagonist - Ligand-based -
Adrenaline uptake inhibitor - Ligand-based -
Aldose reductase inhibitor - Ligand-based -
Anti-Helicobacter pylori - Ligand-based -
Benzodiazepine agonist - Ligand-based -
Benzodiazepine agonist partial - Ligand-based -
Corticotropin releasing factor 1 receptor antagonist - Ligand-based -
Cyclic GMP phosphodiesterase inhibitor - Ligand-based -
Cyclooxygenase inhibitor - Ligand-based -
Dihydroorotate dehydrogenase inhibitor - Ligand-based -
Dihydropteroate synthase inhibitor - Ligand-based -
DNA topoisomerase inhibitor - Ligand-based -
Endothelial growth factor antagonist - Ligand-based -
Excitatory amino acid antagonist - Ligand-based -
Factor VIIa inhibitor - Ligand-based -
Gastrin inhibitor - Ligand-based -
Growth hormone agonist - Ligand-based -
Histamine antagonist - Ligand-based -
Histamine release inhibitor - Ligand-based -
Hsp90 focused library 733 Ligand-basedReceptor-based read more
Interleukin 8 antagonist - Ligand-based -
Irritable Bowel syndrome treatment - Ligand-based -
Kallikrein inhibitor - Ligand-based -
Lactamase C inhibitor - Ligand-based -
Leukotriene B4 antagonist - Ligand-based -
Leukotriene E4 antagonist - Ligand-based -
Lipase inhibitor - Ligand-based -
Lipid peroxidase inhibitor - Ligand-based -
Lipoxygenase inhibitor - Ligand-based -
Liver fibrosis treatment - Ligand-based -
Maillard reaction inhibitor - Ligand-based -
MAO inhibitor - Ligand-based -
Mediator release inhibitor - Ligand-based -
Neurokinin 1 antagonist - Ligand-based -
Neurokinin 3 antagonist - Ligand-based -
Neuropeptide antagonist - Ligand-based -
Neuropeptide Y antagonist - Ligand-based -
Non-steroidal antiinflammatory agent - Ligand-based -
Oxytocin antagonist - Ligand-based -
Para amino benzoic acid antagonist - Ligand-based -
Peroxisome proliferator-activated receptor agonist - Ligand-based -
Peroxisome proliferator-activated receptor gamma agonist - Ligand-based -
Phosphodiesterase inhibitor - Ligand-based -
Phosphodiesterase V inhibitor - Ligand-based -
Phospholipase A2 inhibitor - Ligand-based -
Phospholipase inhibitor - Ligand-based -
Platelet aggregation inhibitor - Ligand-based -
Polarisation inhibitor - Ligand-based -
Potassium channel antagonist - Ligand-based -
Prostaglandin antagonist - Ligand-based -
Prostaglandin synthase inhibitor - Ligand-based -
Protease inhibitor - Ligand-based -
Reverse transcriptase inhibitor - Ligand-based -
Ribonucleoside diphosphate reductase inhibitor - Ligand-based -
Ribonucleoside triphosphate reductase inhibitor - Ligand-based -
Ribonucleotide reductase inhibitor - Ligand-based -
S-adenosyl-L-methionine decarboxylase inhibitor - Ligand-based -
Sigma receptor antagonist - Ligand-based -
Stromelysin inhibitor - Ligand-based -
Substance P antagonist - Ligand-based -
Thromboxane A2 antagonist - Ligand-based -
Thromboxane antagonist - Ligand-based -
Thromboxane synthase inhibitor - Ligand-based -
TNF convertase inhibitor - Ligand-based -
Topoisomerase inhibitor - Ligand-based -
Vanilloid antagonist - Ligand-based -
VLA antagonist - Ligand-based -
Xanthine oxidase inhibitor - Ligand-based -

 

OTAVAchemicals Target-Focused Libraries collection
Name Number
Kinases 67
Proteases 12
GPCRs 25
Ion channels 6
Disease-based libraries 29
Epigenetic targets 7
Protein-Protein Interaction 2
Peptidomimetic 1
Nuclear Receptors 2
Glycomimetic 1
RNA binding 1
General Activities 128
Other 104

 

 

The libraries (SDF, XLS, PDF format) are available on request. Feel free to contact us or use on-line form below to send an inquiry if you are interested to obtain these libraries or if you need more information.

 

 

 

 

 

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