Protein kinases constitute a large family of proteins that is now firmly established as a major class of drug targets for the pharmaceutical industry. With so many inhibitors reported to be in clinical development and many more in preclinical development, kinase inhibitors now make up a significant fraction of most major pharmaceutical companies' pipelines, as well as an area of focus for many biotechnology companies. The increased interest in this class of targets reflects both advances in identifying selective protein kinase inhibitors and a growing perception that these drugs offer a novel, well-tolerated oral therapy in some of the most untreatable cancers.

 

 

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Name	Number of compounds	Approach	Details	Available on-line
1-Phosphatidylinositol-4-phosphate 5-kinase (PIPK) inhibitor	14	Ligand-based	-	search on-line
Abl kinase inhibitor	76	Ligand-based	-	search on-line
Acetate kinase inhibitor	129	Ligand-based	-	search on-line
ADP-thymidine kinase inhibitor	922	Ligand-based	-	search on-line
Aurora kinase inhibitor	364	Ligand-based	-	search on-line
Aurora-B kinase inhibitor	249	Ligand-based	-	search on-line
Aurora-C kinase inhibitor	1162	Ligand-based	-	search on-line
Beta-adrenergic receptor kinase (BARK) inhibitor	1268	Ligand-based	-	search on-line
Check point kinase (CHK) inhibitor	593	Ligand-based	-	search on-line
Cyclin-dependent kinase 1 (CDK1) inhibitor	83	Ligand-based	-	search on-line
Cyclin-dependent kinase 2 (CDK2) inhibitor	905	Ligand-based	-	search on-line
Cyclin-dependent kinase 4 (CDK4) inhibitor	798	Ligand-based	-	search on-line
Cyclin-dependent kinase (CDK) inhibitor	285	Ligand-based	-	search on-line
EphB2 kinase inhibitor	329	Ligand-based	-	search on-line
Epidermal growth factor receptor kinase (EGFR) inhibitor	318	Ligand-based	-	search on-line
Glycogen synthase kinase-3 (GSK3) inhibitor	153	Ligand-based	-	search on-line
G-protein-coupled receptor kinase (GRK) inhibitor	1268	Ligand-based	-	search on-line
Guanidinoacetate kinase inhibitor	254	Ligand-based	-	search on-line
I kappa B kinase 2 (IKK2) inhibitor	347	Ligand-based	-	search on-line
Inositol-trisphosphate 3-kinase (IP3K) inhibitor	78	Ligand-based	-	search on-line
Lombricine kinase inhibitor	163	Ligand-based	-	search on-line
MAP kinase (MAPK) inhibitor	102	Ligand-based	-	search on-line
N-acylmannosamine kinase inhibitor	935	Ligand-based	-	search on-line
NADH kinase inhibitor	871	Ligand-based	-	search on-line
Opheline kinase inhibitor	875	Ligand-based	-	search on-line
Phosphatidylinositol 3-kinase beta (PI3K-C2 beta) inhibitor	1183	Ligand-based	-	search on-line
Phosphatidylinositol 3-kinase gamma (PI3K-C2 gamma) inhibitor	252	Ligand-based	-	search on-line
Phosphoenolpyruvate carboxykinase (PEPCK) inhibitor	26	Ligand-based	-	search on-line
Platelet derived growth factor receptor kinase (PDGFR) inhibitor	1972	Ligand-based	-	search on-line
Protein kinase CK1 inhibitor	1387	Ligand-based	-	search on-line
Protein kinase B (PKB) inhibitor	1030	Ligand-based	-	search on-line
Protein kinase C eta (PKC) inhibitor	16	Ligand-based	-	search on-line
Protein-serine-threonine kinase inhibitor	213	Ligand-based	-	search on-line
Proto-oncogene tyrosine-protein kinase Fyn inhibitor	481	Ligand-based	-	search on-line
Proto-oncogene tyrosine-protein kinase Kit inhibitor	214	Ligand-based	-	search on-line
Pyridoxal kinase inhibitor	5	Ligand-based	-	search on-line
Raf kinase B inhibitor	38	Ligand-based	-	search on-line
Raf kinase inhibitor	74	Ligand-based	-	search on-line
Rho-associated kinase inhibitor	344	Ligand-based	-	search on-line
Ribosomal protein S6 kinase (S6K) inhibitor	10	Ligand-based	-	search on-line
Shikimate kinase inhibitor	453	Ligand-based	-	search on-line
Smooth muscle myosin light chain kinase (MLCK) inhibitor	627	Ligand-based	-	search on-line
Sphinganine kinase inhibitor	244	Ligand-based	-	search on-line
Sphingosine kinase inhibitor	1119	Ligand-based	-	search on-line
Src kinase inhibitor	200	Ligand-based	-	search on-line
Taurocyamine kinase inhibitor	875	Ligand-based	-	search on-line
Thymidine kinase inhibitor	922	Ligand-based	-	search on-line
Tyrosine kinase inhibitor	1147	Ligand-based	-	search on-line
Urokinase inhibitor	21	Ligand-based	-	search on-line
P21-Activated Kinase 1 (PAK1)	2024	Receptor-Based	read more	search on-line
Serine/Threonine-Protein Kinase CHK1 (CHK1)	1946	Receptor-Based	read more	search on-line
Proto-Oncogene Tyrosine-Protein Kinase ABL1	2048	Receptor-Based	read more	search on-line
Extracellular Signal-Regulated Kinase 2 (ERK2)	2053	Receptor-Based	read more	search on-line
Death-Associated Protein Kinase 2 (DAPK-2)	2012	Receptor-Based	read more	search on-line
p38 MAP Kinase Alpha	2221	Receptor-Based	read more	search on-line
Vascular Endothelial Growth Factor Receptor 2 (VEGFR2)	2235	Receptor-Based	read more	search on-line
Aurora B kinase	2069	Receptor-Based	read more	search on-line
Janus Kinase 2 (Jak2)	2190	Receptor-Based	read more	search on-line
Phosphatidylinositol 3-kinase (PI3K)	2040	Receptor-Based	read more	search on-line
3-phosphoinositide-dependent kinase-1 (PDK-1)	1975	Receptor-Based	read more	search on-line
Cyclin Dependent Kinase 2 (CDK2)	1281	Receptor-Based	read more	search on-line
Glycogen Synthase Kinase-3 (GSK3)	980	Receptor-Based	read more	search on-line
Fibroblast growth factor receptor 1 tyrosine kinase (FGFR1K)	1761	Receptor-Based	read more	search on-line
cAMP dependent protein kinase (PKA)	1877	Receptor-Based	read more	search on-line
C-Jun N-Terminal Kinase 2 (Jnk2, Mapk9)	1774	Receptor-Based	-	search on-line
Death-associated protein kinase 1 (DAPK1)	1962	Receptor-Based	-	search on-line
Death-associated protein kinase 3 (DAPK3)	1814	Receptor-Based	-	search on-line

 

 

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